Ultrafastin

Joint pain interferes with normal life. It is capable of overtaking a person at any time and for various reasons. To combat this unpleasant symptom, a wonderful drug, Ultrafastin, was developed. It allows you to quickly remove pain and excessive inflammation.

Indications Ultrafastin

The main function of Ultrafastin is to provide anti-inflammatory and analgesic effects. The joints and muscles of a person can start to worry at any time. This is due to excessive exposure to them through means of increased physical work. Suffering tendons and muscles may be due to severe trauma. Therefore, the main indications for the use of Ultrafastin are post-traumatic pains.

The drug is applied externally, which facilitates the whole situation. You can take it with you and use it at any time. The effectiveness of Ultrafastin has been proven not by one year of trials. Ultrafastin really helps to cope with even the most severe pain and eliminates an unpleasant symptom in a matter of minutes.

Despite its safety, it should not be used without the knowledge of the doctor. After all, the medicine can lead to the development of adverse reactions. Concerning this topic we will discuss below. 

Release form

Ultrafastin is available as a gel for external use. In fact, this form of output is very convenient. You can carry the medicine with you, because the weight of the tuba does not exceed 30 grams. There is a larger package, it contains a medicine with a volume of 50 grams. The concentration of the active component is 2.5%. By the way, the main substance is ketoprofen lazine salt.

The auxiliary components of Ultrafastin does not contain and therefore is the safest among others. Ketoprofen lazine salt helps a person cope with the pain of any localization. It is enough simply to apply the gel to the affected area and the pain syndrome will begin to recede. To achieve a special therapeutic effect, it is necessary to follow the recommendations of the doctor.

It is worth noting that the drug has no other forms of release. In fact, this is very important information. It will avoid getting on fakes. 

[1]

Pharmacodynamics

The main active ingredient of Ultrafastin is ketoprofen. It has a pronounced analgesic and anti-inflammatory effect. The main component is able to reduce the activity of cyclooxygenase-1 and cyclooxygenase-2. This leads to a decrease in the production of prostaglandins, and in fact they play a major role in the pathogenesis of the pain syndrome. This is the pharmacodynamics of the drug, but that's not all.

The mechanism of anti-inflammatory effect has not been fully studied. It is known that ketoprofen leads to difficulties in the release of lysosomal enzymes. In addition, it significantly reduces the oxygen metabolism of neutrophilic cells. The drug actively slows the migration of macrophages and thus leads to a decrease in the activity of the bradykinin system. All these actions lead to a reduction in phase II inflammation. This is due to a reduced migration of granulocytes and macrophages into the synovial membrane. All this leads to the formation of cellular filtrates. 

[2]

Pharmacokinetics

The components of Ultrafastin perfectly penetrate the skin. Thus, there is an analgesic and anti-inflammatory effect. And you can feel relief almost immediately. The basis of pharmacokinetics is the rate of absorption and distribution. In this case, these parameters completely depend on the thickness of the skin. A special role here is played by the thickness of the subcutaneous fat layer, as well as the intensity of the blood supply at the site of the lesion.

With external use of Ultrafastin, its maximum amount in the blood plasma is observed after an hour. Virtually 99% of the main absorbed component interacts with blood plasma proteins.

As for bioavailability, it is 5%. The effect of the first origin is observed in the liver. The drug is completely excreted in the urine, 80% in the form of metabolites and 10% unchanged. Even if Ultravastine is used for a long time, it is not able to accumulate in the body. 

[3], [4], [5]

Dosing and administration

The remedy is used exclusively externally. The gel must be applied to the affected area with a thick layer and rubbed with light massaging movements. This will speed up the process of absorption and, accordingly, of relief. In general, the method of administration and dose should be prescribed by a doctor, depending on the severity of the inflammatory and painful process.

Ultrafastin should be used 2-3 times a day, this will achieve maximum therapeutic effect. The duration of treatment is determined on an individual basis. Only a specialist can make this decision. Self-use means is not recommended.

The gel has no odor, which allows it to be applied anywhere. Moreover, it leaves no oily traces and is perfectly absorbed through the skin. The agent does not contain dyes in its composition. All this suggests that it is possible to use Ultrafastin without the help of a dry bandage. 

[8]

Use Ultrafastin during pregnancy

Medication is not used orally, so there can be no contraindications. But, despite this use of the gel during pregnancy is prohibited in the third trimester.

Most often, drugs should not be taken in the early stages of pregnancy. In this case, everything is somewhat different. This is due to the fact that the medicine is able to affect the mother's body. Despite the fact that in the third trimester the use is not prohibited, it should be done only with the permission of the doctor. After all, as described above, the mechanism of action of ketoprofen was not thoroughly studied. Therefore, the risk of unfavorable consequences persists.

In general, the medication penetrates exclusively into the subcutaneous layers. But, nevertheless, it is concentrated in the blood plasma. How this can affect the baby's future is not known. Therefore, you should not experiment with this. Any drug is taken only if the positive result for the mother is much higher than the possible complications for the baby. 

Contraindications

The main contraindication is the presence of hypersensitivity in humans. Many people ignore this recommendation. The use of the drug in hypersensitivity is fraught with the development of serious allergic reactions from the body. Another contraindication to use is the presence of an open wound. Apply gel to such a site is prohibited.

Use the medication is not possible with eczema, as well as with wet dermatoses. The presence of infected abrasions and infectious lesions of the skin also refers to a number of contraindications. Apply gel is not recommended in the presence of burns and wounds. In this case, the gel can lead to an increase in the already existing symptoms. Such an effect will adversely affect the existing wound.

Due to its features and strong active ingredient, it is not necessary to use the product for children under 15 years of age. Compliance with these recommendations will not exacerbate the situation. 

[6]

Side effects Ultrafastin

The organism rarely responds negatively to such an effect. As a result of the research, it was revealed that side effects are not common. Sometimes allergic reaction from the skin can develop. It is characterized by the appearance of itching, redness and rash. To develop, is capable of skin eczema, purpura and photosensitization.

Very rarely the skin becomes too sensitive to bright light. This condition is characterized by the appearance of severe papular exanthema. This disease is not pleasant and is prone to recurrence.

Ketoprofen is capable of provoking bronchospasm in those patients who are too sensitive to the use of acetylsalicylic acid. The frequency of side effects, as well as their manifestation, depend on the area of the treated area and the amount of the agent applied. When using a bandage, other symptoms can also be documented. Including deviations from the work of the kidneys and the gastrointestinal tract. 

[7]

Overdose

There were no cases of strange reactions on the part of the body during the period of application of the remedy. In general, Ultrafastin does not cause an overdose, but exclude the possibility of its appearance is not necessary. If the gel is applied excessively to the skin, severe allergic reactions may develop. Moreover, the systematic use of the agent in large quantities and not in a small area of the skin can lead to the development of deviations from the gastrointestinal tract and kidneys.

The gel can be swallowed casually. Situations are different and this should not be completely ruled out. Such an effect on the body can lead to the development of serious poisoning. Therefore, if the product gets inside, you should immediately rinse the stomach. After all, the consequences can be really heavy. After that, it is worth informing the doctor about the situation and, if necessary, starting symptomatic therapy. 

[9]

Interactions with other drugs

Negative reactions with the use of several drugs can appear simultaneously. This is possible, but only if Ultrastatin is used for a long time. Thus, simultaneous interaction with other drugs, including heparins, can lead to the development of bleeding. A similar action can occur in the case of oral anticoagulants, thrombolytic agents and cefoperazone

Ultravastin can reduce the effect of diuretics. As for oral hypoglycemic drugs, as well as insulin, it is possible to strengthen the effect of the latter. Therefore, if you need to share these funds, you need to correctly adjust the dose. This question should be solved together with the attending physician.

The use of Ultrafastin along with sodium valproate may result in impaired platelet aggregation. In addition, it is possible to increase the content of nifedipine and verapamil in blood plasma. The agent can lead to an increase in the action of methotrexate. It is highly not recommended to use the gel together with acetylsalicylic acid. Ultrafastin does not accept alcohol. Perhaps strengthening its effect on the body.

[10], [11], [12], [13], [14],

Storage conditions

The first thing to do is to store ultravastin away from the light. The fact is that drugs can deteriorate under the influence of bright sunlight. So the best place is where it's dark. Another important condition of storage is the exclusion of moisture. The fact is that many drugs can get wet. This will lead to the fact that they will deteriorate. Therefore, it is better to choose a dry place, the bathroom is definitely not the best option.

Do not keep the tube open. This will result in the absorption or volatilization of substances. There may be a reaction with air. Therefore, the bottle must be permanently closed. Tightness is an important condition for any storage.

Observe the necessary and optimal temperature. It is desirable that the gel is at room temperature, in a dark place that does not undergo heating. For this product, the optimal temperature conditions are 15-25 degrees Celsius. Finally, drugs should be kept away from children. This will save them from consuming Ultrafastin. 

[15]

Shelf life

Use an overdue means in any case impossible. This can lead to poisoning. In most cases, the pharmacological action is weakened by the end of the shelf life. Therefore, the use of the gel will not give any result. So, the shelf life of this gel is 2 years. At the end of a given period, it is worth to get rid of it.

It is desirable to carry out an audit of medicines more often. This will allow timely elimination of those drugs that you can not use anyway. Overdue gel is a combination of substances that have unpredictable effects. They can cause serious harm to the human body.

During the whole period, you need to monitor the appearance of the gel. He should not change his consistency, color and smell. If this happens, then the recommended storage conditions have not been met, which has resulted in damage to the product. Therefore, to monitor the condition of the gel is mandatory. Only this way you can protect your own health.