Sulfocamfocaine

Sulfocamfocaine is a medicine that contains two active ingredients: procaine and sulfocamphoric acid. Here is brief information about each of them:

1. Procaine: It is a local anesthetic that blocks the conduction of nerve impulses and temporarily reduces sensitivity to pain in the area of application. Procaine is widely used in medicine for anesthesia in minimally invasive procedures and manipulations such as injections, dental procedures and others.
2. Sulfocamphoric acid: This component has antiseptic and anti-inflammatory properties. It helps to reduce inflammation and the risk of infection in the area where the medicine is applied.

Sulfocamfocaine is commonly used for local anesthesia in a variety of medical procedures, including injections, dental procedures, wound care, and burns. It can be used as a solution for injection, ointments or gels for external application.

It is important to remember that the use of sulfocamfocaine should be supervised and recommended by a medical professional to avoid possible side effects and complications.

Indications Sulfocamfocaine

1. Local anesthesia: Used for temporary anesthesia in the area of application. This may include injections into the skin, mucous membranes, or local anesthetic procedures.
2. Dental procedures: Sulfocamfocaine may be used for anesthesia in dental procedures such as tooth extraction, treatment of tooth decay, or other dental interventions.
3. Procedures in minimally invasive surgery: Can be used for anesthesia in minimally invasive surgical procedures such as local injections or diagnostic puncture procedures.
4. Treatment of wounds and burns: Used for anesthesia and antiseptic treatment of wounds, burns and other skin injuries.
5. Cosmetic procedures: Used for anesthesiain cosmetic procedures such as injections of dermal fillers or botulinum toxin.

Release form

1. Solution for injection

• Description: Sulfocamfocaine is most commonly available as a solution for injection, which can be used for intramuscular (IM) or subcutaneous (SC) administration.
• Concentrations: The solution for injection usually contains a certain ratio of procaine to sulfocamphoric acid, e.g., 0.5% procaine to 2% sulfocamphoric acid.
• Packaging: The solution is usually packaged in ampoules of 1, 2 or 5 ml.

2. Gel or ointment for external application

• Description: Although more rare, sulfocamfocaine may be available in the form of a gel or ointment for external application. This form is applied directly to the skin in the area of pain or inflammation.
• Concentrations and Packaging: Details of active ingredient concentrations and packaging types may vary by manufacturer and regional standards.

Pharmacodynamics

Sulfocamfocaine is a combination of two active ingredients: procaine (local anesthetic) and sulfocamphoric acid. Procaine blocks the conduction of nerve impulses, causing temporary loss of sensation in the area of application, while sulfocamphoric acid provides antimicrobial action.

Sulfocamfocaine is used for pain relief in medical procedures such as infiltration anesthesia and blockages. It has analgesic and antimicrobial effects, making it useful in the treatment of skin and soft tissue infections.

Dosing and administration

Ways of application:

Sulfocamfocaine is usually available as a solution for injection. These are solutions that are administered subcutaneously, intramuscularly, and sometimes intravenously depending on the medical indication.

Injection application:

1. Subcutaneous injection (P/k):

   • Used for local anesthesia in minor surgical procedures or in dentistry.
   • The dosage is usually 1 to 2 mL of solution.

2. Intramuscular injection (IM):

   • It is used to achieve a faster and more intense analgesic effect.
   • The dosage may vary from 1 to 5 ml depending on the severity of the pain syndrome and the anatomical area.

3. Intravenous (I/V):

   • Usually used in emergencies for instant anesthesia.
   • The dosage is strictly controlled and should be administered by medical professionals.

Dosage:

• Theinitial adultdose is usually 1-2 mL of solution, which may be repeated depending on clinical need and patient tolerability.
• Themaximum daily dose should not exceed 10 mL, as high doses may result in an increased risk of side effects, including systemic reactions to procaine and sulfocamphoric acid.

Special Instructions:

• Patient monitoring: It is important to monitor the patient for reactions to the drug, especially if intravenous administration is used.
• Use in specialized settings: Injections should be administered by medical professionals with appropriate training and experience with injectable anesthetics.
• Allergic reactions: It is necessary to take into account the possible allergy of the patient to the components of the drug, especially procaine.
• Adherence to asepsis and antisepsis: It is important to strictly follow the rules of asepsis and antisepsis when administering injections to prevent infectious complications.

Use Sulfocamfocaine during pregnancy

The use of sulfocamfocaine during pregnancy may require special attention and doctor's recommendations. Generally, the use of the medication is avoided during pregnancy, especially in the first trimester when the baby's organs and systems are actively forming.

Before using sulfocamfocaine or any other drug during pregnancy, it is important to discuss it with your doctor. Your doctor can assess the potential risks and benefits of the drug in your particular situation and make an informed decision about its use.

Contraindications

1. Hypersensitivity: People with known hypersensitivity to procaine, sulfocamphoric acid, or other amide anesthetics should not use this drug because of the risk of allergic reactions, including anaphylaxis.
2. Pregnancy and breastfeeding: The use of sulfocamfocaine during pregnancy may be undesirable or contraindicated due to insufficient information on its safety for the fetus. In addition, the drug may pass into breast milk and cause undesirable effects in the infant.
3. Skin lesions: The drug should be avoided in the presence of skin lesions, burns, infected wounds or other skin conditions, as it may aggravate the condition and cause irritation.
4. High blood pressure: In people with high blood pressure, caution should be exercised when using sulfocamfocaine because of its ability to produce an excitatory effect on the central nervous system and increase blood pressure.
5. Cardiovascular disease: Patients with cardiovascular disease, such as arrhythmias or ischemic heart disease, should use sulfocamfocaine with caution because of its possible adverse effects on the cardiovascular system.
6. Diabetes mellitus: In patients with diabetes mellitus, caution should be exercised when using sulfocamfocaine because of its ability to raise blood glucose levels.
7. Central nervous system diseases: Sulfocamfocaine should be used with caution in patients with central nervous system diseases such as epilepsy or nerve impulse conduction disorders due to the possibility of worsening symptoms.
8. Children: The use of sulfocamfocaine in children may require special caution and should be administered under medical supervision.
9. Elderlypatients: The elderly may be more sensitive to the effects of sulfocamfocaine, so it should be used with caution.

Side effects Sulfocamfocaine

1. Allergic reactions: It is possible to develop allergic reactions to the components of the drug, manifested as itching, skin rash, swelling or redness at the site of application.
2. Systemic Reactions: Systemic reactions such as dizziness, pallor, feeling of warmth or cold sweat may occur when the drug is used as an injection.
3. Local reactions: Local reactions may occur at the injection site, such as redness, swelling, soreness, or a small hematoma.
4. Tissue necrosis: Complications in the form oftissue necrosis or ulceration may develop if the drug is used as an injection or overused.
5. Nervous system disorders: In rare cases, nervous system disorders such as headache, tinnitus, seizures or paralysis may occur.
6. Otherside effects: Other rare side effects may occur, including abnormal heart rhythm, arterial hypertension, or arterial hypotension.

Overdose

1. Dizziness and drowsiness.
2. Speech queues and difficulty in pronouncing words.
3. Tremors and muscle cramps.
4. Increased heartbeat and arrhythmias.
5. Pulmonary edema and bronchospasm.

Interactions with other drugs

1. Other local anesthetics: The use of sulfocamfocaine together with other local anesthetics may result in a stronger anesthetic effect. This may increase the risk of systemic side effects such as toxic reactions on the heart or central nervous system.
2. Vasoconstrictor drugs: The use of sulfocamfocaine with drugs that have a vasoconstrictor effect, such as adrenaline or norepinephrine, may result in longer duration and greater anesthetic effect due to delayed absorption.
3. Drugs affecting the systemic circulation: Interaction of sulfocamfocaine with drugs affecting the systemic circulation, such as antiarrhythmic drugs or beta-adrenoblockers, may increase or decrease their effects due to possible influence on absorption or metabolism.
4. Drugs affecting the CNS: The use of sulfocamfocaine together with drugs affecting the central nervous system, such as sedatives or antidepressants, may increase their depressant effect on the CNS.
5. Drugs causing metabolic effects: Sulfocamfocaine may interact with drugs that cause metabolic changes, such as liver enzyme inhibitors or inducers, which may alter the rate of metabolism and excretion of sulfocamfocaine from the body.